发明名称 BICYCLOAMINE DERIVATIVE
摘要 <p>Compounds represented by formula (I) and pharmaceutically acceptable salts thereof have excellent sodium channel inhibitory action and are useful as therapeutic agents and analgesics for various kinds of neuralgia, neuropathy, epilepsy, insomnia, premature ejaculation and the like. wherein Q represents ethylene, etc., R 1 , R 2 and R 3 represent hydrogen, etc., X 1 represents C 1-6 alkylene, etc., X 2 represents C 1-6 alkylene, etc., A 1 represents a 5- to 6-membered heterocyclic group, etc., and A 2 represents C 6-14 aryl, etc.</p>
申请公布号 EP2241567(A1) 申请公布日期 2010.10.20
申请号 EP20090710649 申请日期 2009.02.09
申请人 EISAI R&D MANAGEMENT CO., LTD. 发明人 OZAKI, FUMIHIRO;SOEJIMA, MOTOHIRO;ISHIDA, TASUKU;NORIMINE, YOSHIHIKO;KURUSU, NOBUYUKI;DOI, ERIKO;KANEKO, TOSHIHIKO;HASEGAWA, DAIJU;KOBAYASHI, KIYOAKI;YAMAMOTO, NOBORU
分类号 C07D451/06;A61K31/439;A61K31/46;A61K31/4985;A61K31/53;A61K31/5377;A61K31/5383;A61K31/55;A61P3/12;A61P15/00;A61P25/00;A61P25/04;A61P25/08;A61P25/20;A61P29/02;A61P43/00;C07D451/14;C07D519/00 主分类号 C07D451/06
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