发明名称 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL TERTIARY-HETEROALKYLAMINES USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY
摘要 The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer protein-I) and compounds, compositions and methods for treating atherosclerosis and other coronary artery diseases.
申请公布号 CA2345118(C) 申请公布日期 2010.04.27
申请号 CA19992345118 申请日期 1999.09.23
申请人 MONSANTO COMPANY 发明人 SIKORSKI, JAMES A.;DURLEY, RICHARD C.;MISCHKE, DEBORAH A.;REINHARD, EMILY J.;FOBIAN, YVETTE M.;TOLLEFSON, MICHAEL B.;WANG, LIJUAN;GRAPPERHAUS, MARGARET L.;HICKORY, BRIAN S.;MASSA, MARK A.;NORTON, MONICA B.;VERNIER, WILLIAM F.;PARNAS, BARRY L.;PROMO, MICHELE A.;HAMME, ASHTON T.;SPANGLER, DALE P.;RUEPPEL, MELVIN L.
分类号 C07C215/16;C07D251/46;A61K31/135;A61K31/136;A61K31/137;A61K31/16;A61K31/17;A61K31/196;A61K31/245;A61K31/277;A61K31/33;A61K31/341;A61K31/381;A61K31/395;A61K31/40;A61K31/403;A61K31/404;A61K31/4045;A61K31/42;A61K31/421;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4412;A61K31/4418;A61K31/4453;A61K31/472;A61K31/496;A61K31/505;A61K31/53;A61P3/06;A61P9/10;A61P43/00;B01J31/12;C07B57/00;C07B61/00;C07C213/04;C07C215/08;C07C215/50;C07C215/68;C07C215/76;C07C217/58;C07C217/84;C07C217/86;C07C217/88;C07C217/90;C07C219/34;C07C225/22;C07C229/60;C07C233/65;C07C233/69;C07C233/80;C07C235/38;C07C235/56;C07C237/30;C07C237/38;C07C239/20;C07C255/54;C07C255/55;C07C255/58;C07C275/34;C07C275/40;C07C291/04;C07C311/04;C07C311/08;C07C311/21;C07C311/24;C07C311/60;C07C317/32;C07C317/36;C07C319/20;C07C323/19;C07C323/25;C07C323/31;C07C323/32;C07C323/36;C07C323/37;C07C323/44;C07C323/65;C07D207/32;C07D207/323;C07D207/335;C07D209/08;C07D209/32;C07D209/86;C07D213/26;C07D213/30;C07D213/38;C07D213/64;C07D213/643;C07D213/65;C07D213/66;C07D213/85;C07D217/24;C07D225/08;C07D239/26;C07D239/34;C07D251/16;C07D251/42;C07D257/04;C07D263/06;C07D295/135;C07D295/192;C07D307/14;C07D307/42;C07D307/52;C07D309/12;C07D333/20;C07D333/28;C07F7/18 主分类号 C07C215/16
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