发明名称 |
NILOTINIB INTERMEDIATES AND PREPARATION THEREOF |
摘要 |
Intermediates of Nilotinib were prepared, including, for example, 3-(trifluoromethyl-5-(4-methyl-1H-imidazole-1-yl)-benzeneamine; 3-(4-(pyridin-3-yl)pyrimidin-2-ylamino) -4-methylbenzoyl halogen dihydrochloride; and N-(3-Bromo-5-trifluoromethylphenyl)-4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzamide. Nilotinib.3HCl and its crystalline forms are also described.
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申请公布号 |
US2010016590(A1) |
申请公布日期 |
2010.01.21 |
申请号 |
US20090505213 |
申请日期 |
2009.07.17 |
申请人 |
TEVA PHARMACEUTICAL INDUSTRIES LTD. |
发明人 |
WANG YANLING;LI JIE;KANSAL VINOD KUMAR;ZHU JIRANG;LIFSHITZ-LIRON REVITAL;MISTRY DHIRENKUMAR N.;VASOYA SANJAY L.;ARIYAMUTHU SUNDARASELVAN;PILARSKI GIDEON;HE XUNGUI |
分类号 |
C07D401/14;C07D233/56;C07D401/04 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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地址 |
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