发明名称 SALTS OF (R)-5-(2-PHENYLSULPHONYLETHENYL)-3-(N- METHYLPYRROLIDIN-2-YLMETHYL)-1H-INDOLE, 5-BROMO-3-[(R)-1- METHYL-PYRROLIDIN-2- YLMETHYL]-1H-INDOLE AND OF ELETRIPTAN
摘要 The present invention relates to salts of (R)-5-(2-phenylsulphonylethenyl)-3-(N- methylpyrrolidin-2-ylmethyl)-lH-indole of the Formula:(I) wherein HX is an acid selected from para-toluene sulfonic acid, benzene sulphonic acid, trifluoroacetic acid, methane sulphonic acid, formic acid and succinic acid; and to processes of preparing and using such salts.
申请公布号 WO2009142771(A3) 申请公布日期 2010.01.14
申请号 WO2009US03190 申请日期 2009.05.22
申请人 PLUS CHEMICALS, S.A.;TEVA PHARMACEUTICALS USA, INC.;KANSAL, VINOD, KUMAR;MISTRY, DHIRENKUMAR, N.;PATEL, RAKESH, RAVJIBHAI;GUPTA, PRIYANKA 发明人 KANSAL, VINOD, KUMAR;MISTRY, DHIRENKUMAR, N.;PATEL, RAKESH, RAVJIBHAI;GUPTA, PRIYANKA
分类号 C07D403/06;A61K31/404 主分类号 C07D403/06
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