发明名称 NOVEL NITROGENATED HETEROCYCLIC COMPOUND AND SALT THEREOF
摘要 <p>A nitrogen-containing heterocyclic compound represented by the general formula: wherein the dashed line represents a single bond or a double bond; R 1 , R 2 , R 3 , R 4 and R 5 independently represent a hydrogen atom, halogen atom, a lower alkyl, aryl, lower alkoxy or monocyclic heterocyclic group which may be substituted or the like; R 6 represents a lower alkyl, aryl, monocyclic heterocyclic, bicyclic heterocyclic or tricyclic heterocyclic group which may be substituted; X 1 represents a lower alkylene group or the like; X 2 represents a lower alkylene, lower alkenylene or lower alkynylene group which may be substituted; X 3 represents an oxygen atom, sulfur atom, a sulfinyl group, sulfonyl group or the like; Y 1 represents a bivalent cyclic group, containing a nitrogen, which may be substituted or the like; and Z 1 represents a nitrogen atom, a carbon atom which may be substituted or the like, or a salt thereof. The compound or salt has a potent antibacterial activity and a high safety, and is therefore useful as an excellent antibacterial agent.</p>
申请公布号 EP1900732(A4) 申请公布日期 2009.11.18
申请号 EP20060767173 申请日期 2006.06.22
申请人 TOYAMA CHEMICAL CO., LTD.;TAISHO PHARMACEUTICAL CO., LTD 发明人 KIYOTO, TARO;TANAKA, TADASHI;TSUTSUI, YASUHIRO;ANDO, JUNICHI;MOTONO, MAI;KAWAGUCHI, YASUKO;NOGUCHI, TOSHIYA;USHIKI, YASUNOBU;USHIYAMA, FUMIHITO;URABE, HIROKI
分类号 C07D401/06;A61K31/4709;A61K31/496;A61P31/04;C07D401/14;C07D405/14;C07D409/14;C07D491/056 主分类号 C07D401/06
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