PROCESS FOR PREPARING CRYSTALLINE CALCIUM MUPIROCIN DIHYDRATE
摘要
<p>Provided herein are methods of preparing crystalline mupirocin calcium dihydrate comprising combining solid mupirocin, solid calcium carbonate, and water in an amount sufficient to form a heterogeneous mixture and precipitate crystalline mupirocin calcium dihydrate from the mixture. In some embodiments, the methods produce nanocrystalline mupirocin calcium dihydrate, suitable for use in pharmaceutical formulations.</p>
申请公布号
WO2009092991(A1)
申请公布日期
2009.07.30
申请号
WO2008GB04307
申请日期
2008.12.30
申请人
PLIVA HRVATSKA D.O.O.;BUCKS, TERESA, ANNE;DEFTERDAROVIC, NAFIS;TUDJA, MARIJAN;CAVUZIC, DRAZEN