发明名称 |
PROCESS FOR THE PREPARATION OF PYRAZOLYLAMINOQUINAZOLINE DERIVATIVES COMPRISING A PHOSPHATE GROUP |
摘要 |
<p>The invention relates to a new process useful in the preparation of pharmaceutical compounds such as 2-{ethyl[3-({4-[(5-{2-[(3-fluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl) amino]quinazolin-7-yl}oxy)propyl]amino}ethyl dihydrogen phosphate (AZD1152) and intermediates used therein.</p> |
申请公布号 |
KR20090008450(A) |
申请公布日期 |
2009.01.21 |
申请号 |
KR20087029568 |
申请日期 |
2007.05.14 |
申请人 |
ASTRAZENECA AB |
发明人 |
PITTAM JOHN DAVID;SEPENDA GEORGE JOSEPH |
分类号 |
C07D239/94;C07F9/02 |
主分类号 |
C07D239/94 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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