发明名称 SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-PYRIDO[4,3-B]INDOLES, METHODS FOR THE PRODUCTION AND USE THEREOF
摘要 The invention relates to antagonists of 5-HT<SUB>6 </SUB>serotonin<SUB/>receptors which simultaneously control the homeostasis of calcium ions in cells and is in the form of substituted 2,3,4,5-tetrahydro-1h-pyrido[4,3-b]indoles of general formula (1), wherein R<SUP>1</SUP> is an aminogroup substituent selected form optionally substituted C<SUB>1</SUB>-C<SUB>5</SUB> alkyl; R<SUP>2</SUP> <SUB>i</SUB>
申请公布号 WO2008123796(A2) 申请公布日期 2008.10.16
申请号 WO2008RU00196 申请日期 2008.04.01
申请人 ALLA CHEM, LLC;IVASHCHENKO, ANDREY ALEXANDROVICH;IVASHCHENKO, ALEXANDER VASILIEVICH;TKACHENKO, SERGEY YEVGENIEVICH;FROLOV, YEVGENIY BORISOVICH;MITKIN, OLEG DMITRIEVICH;KRAVCHENKO, DMITRI VLADIMIROVICH;OKUN, ILYA MATUSOVICH;SAVCHUK, NIKOLAY FILIPPOVICH 发明人 IVASHCHENKO, ANDREY ALEXANDROVICH;IVASHCHENKO, ALEXANDER VASILIEVICH;TKACHENKO, SERGEY YEVGENIEVICH;FROLOV, YEVGENIY BORISOVICH;MITKIN, OLEG DMITRIEVICH;KRAVCHENKO, DMITRI VLADIMIROVICH;OKUN, ILYA MATUSOVICH;SAVCHUK, NIKOLAY FILIPPOVICH
分类号 C07D471/04;A61K31/437;A61P37/02;A61P37/08 主分类号 C07D471/04
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