摘要 |
The invention relates to antagonists of 5-HT<SUB>6 </SUB>serotonin<SUB/>receptors which simultaneously control the homeostasis of calcium ions in cells and is in the form of substituted 2,3,4,5-tetrahydro-1h-pyrido[4,3-b]indoles of general formula (1), wherein R<SUP>1</SUP> is an aminogroup substituent selected form optionally substituted C<SUB>1</SUB>-C<SUB>5</SUB> alkyl; R<SUP>2</SUP> <SUB>i</SUB> |
申请人 |
ALLA CHEM, LLC;IVASHCHENKO, ANDREY ALEXANDROVICH;IVASHCHENKO, ALEXANDER VASILIEVICH;TKACHENKO, SERGEY YEVGENIEVICH;FROLOV, YEVGENIY BORISOVICH;MITKIN, OLEG DMITRIEVICH;KRAVCHENKO, DMITRI VLADIMIROVICH;OKUN, ILYA MATUSOVICH;SAVCHUK, NIKOLAY FILIPPOVICH |
发明人 |
IVASHCHENKO, ANDREY ALEXANDROVICH;IVASHCHENKO, ALEXANDER VASILIEVICH;TKACHENKO, SERGEY YEVGENIEVICH;FROLOV, YEVGENIY BORISOVICH;MITKIN, OLEG DMITRIEVICH;KRAVCHENKO, DMITRI VLADIMIROVICH;OKUN, ILYA MATUSOVICH;SAVCHUK, NIKOLAY FILIPPOVICH |