发明名称 Compounds Useful In Therapy
摘要 Compounds of formula (I), or pharmaceutically acceptable derivatives thereof, wherein: R<SUP>1 </SUP>represents a group selected from H, CF<SUB>3</SUB>, and C<SUB>1-6 </SUB>alkyl (optionally substituted by C<SUB>1-6 </SUB>alkyloxy or triazolyl); R<SUP>2 </SUP>represents halo; Ring A represents a 5- or 6-membered heterocyclic ring containing at least one N atom (the ring being optionally bridged with two or more carbon atoms); R<SUP>3 </SUP>represents a 5- or 6-membered heterocyclic ring containing at least one atom selected from N, O or S, the heterocyclic ring being optionally substituted by one or more groups selected from C<SUB>1-6 </SUB>alkyl oxo or NH<SUB>2</SUB>, the heterocyclic ring being further optionally fused to a 5- or 6-membered aryl or heterocyclic ring containing at least one atom selected from N, O or S, the fused aryl or heterocyclic ring being substituted by one or more halo atoms; are useful for treating a disorder for which a V1a antagonist is indicated, in particular, dysmenorrhea.
申请公布号 US2008188478(A1) 申请公布日期 2008.08.07
申请号 US20060912592 申请日期 2006.04.18
申请人 PFIZER INC. 发明人 BRYANS JUSTIN STEPHEN;BUNNAGE MARK EDWARD;JOHNSON PATRICK STEPHEN;MASON HELEN JANET;ROBERTS LEE RICHARD;RYCKMANS THOMAS;STOBIE ALAN;UNDERWOOD TOBY JAMES
分类号 A61K31/454;A61K31/437;A61K31/5025;A61P25/00;C07D401/04;C07D471/04;C07D487/04 主分类号 A61K31/454
代理机构 代理人
主权项
地址
您可能感兴趣的专利