PROCESS FOR THE PREPARATION OF 6-ALPHA, 9-ALPHA-DIFLUORO-17-ALPHA - ((2-FURANYLCARBONYL)OXY)-11-BETA -HYDROXY-16-ALPHA -METHYL-S-OXO-ANDROSTA-1,4-DIENE-17-BETA- -CARBOTHIOIC ACID S-FLUOROMETHYL
摘要
A novel process for preparing a compound of formula (I), which comprises converting a compound of formula (II) to a compound of formula (I) via a compound of formula (III), or a salt thereof (III), without isolating any intermediates.
申请公布号
WO2007144363(A3)
申请公布日期
2008.05.02
申请号
WO2007EP55805
申请日期
2007.06.13
申请人
GLAXO GROUP LIMITED;BERRY, MALCOLM, BRIAN;HUGHES, MARK, JASON;PARRY-JONES, DAVID;SKITTRALL, STEPHEN, JOHN
发明人
BERRY, MALCOLM, BRIAN;HUGHES, MARK, JASON;PARRY-JONES, DAVID;SKITTRALL, STEPHEN, JOHN