| 发明名称 |
6H-THIENO[2,3-b]PYRROLE DERIVATIVES AS ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE (GNRH) |
| 摘要 |
The invention relates to a group of novel thieno-pyrrole compounds of Formula (I): wherein: R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4 </SUP>and R<SUP>5 </SUP>are as defined in the specification, which are useful as gonadotrophin releasing hormone antagonists. The invention also relates to pharmaceutical formulations of said compounds, methods of treatment using said compounds and to processes for the preparation of said compounds.
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| 申请公布号 |
US2008045517(A1) |
申请公布日期 |
2008.02.21 |
| 申请号 |
US20070752007 |
申请日期 |
2007.05.22 |
| 申请人 |
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发明人 |
FOOTE KEVIN M.;MATUSIAK ZBIGNIEW;DOSSETTER ALEXANDER G.;ARNOULD JEAN CLAUDE;LAMORLETTE MARYANNICK A.;DELOUVRIE BENEDICTE;HAMON ANNIE |
| 分类号 |
A61K31/541;A61K31/407;A61K31/44;A61K31/445;A61K31/496;A61K31/506;A61K31/5377;A61P35/00;C07D213/02;C07D221/00;C07D239/24;C07D277/02;C07D279/10;C07D295/00 |
主分类号 |
A61K31/541 |
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