发明名称 SUBSTITUTED UREAS
摘要 <p>Urea derivatives having excellent DGAT inhibiting activity or pharmacologically acceptable salts thereof, namely, urea derivatives represented by the general formula (I) or pharmacologically acceptable salts thereof: (I) wherein R&lt;SUP&gt;1&lt;/SUP&gt; is C&lt;SUB&gt;6-10&lt;/SUB&gt; aryl which may be substituted with one member selected from group (a) of substituents and/or one to four members independently selected from group (b) of substituents, or the like; R&lt;SUP&gt;2&lt;/SUP&gt; is C&lt;SUB&gt;6-10&lt;/SUB&gt; aryl which may be substituted with one member selected from group (a) of substituents and/or one to four members independently selected from group (b) of substituents, or the like; R&lt;SUP&gt;3&lt;/SUP&gt; and R&lt;SUP&gt;4&lt;/SUP&gt; are each independently hydrogen or the like; A is C&lt;SUB&gt;2-4&lt;/SUB&gt; alkylene wherein one of the methylene groups constituting the main chain may be replaced by vinylene, oxygen, sulfur, sulfinyl, or sulfonyl, or the like; Q is -N(Me)- or sulfur; T is =CH- or nitrogen; and U and V are each independently =CH- or the like.</p>
申请公布号 WO2006019020(A1) 申请公布日期 2006.02.23
申请号 WO2005JP14633 申请日期 2005.08.10
申请人 SANKYO COMPANY, LIMITED;HAYAKAWA, ICHIRO;YOSHIDA, MASAO;SUGANO, YUICHI;KURATA, HITOSHI;TANIMOTO, TATSUO;KARASAWA, HIROSHI;KOHAMA, TAKAFUMI;UTO, YOSHIKAZU 发明人 HAYAKAWA, ICHIRO;YOSHIDA, MASAO;SUGANO, YUICHI;KURATA, HITOSHI;TANIMOTO, TATSUO;KARASAWA, HIROSHI;KOHAMA, TAKAFUMI;UTO, YOSHIKAZU
分类号 (IPC1-7):C07D233/64;C07D413/12;A61K31/416;C07D405/12;C07D403/06;C07D401/14;C07D401/06;C07D401/04;C07D285/12;C07D277/28;C07D249/12;C07D249/08;A61P43/00;A61P29/00;A61P27/02;A61P25/02;A61P19/06;A61P19/02;A61P15/00;A61P13/12;A61P11/00;A61P9/12;A61P9/10;A61P3/10;A61P3/06;A61P3/04;A61P1/16;A61K31/443;A61K31/433;A61K31/426;A61K31/422;A61K31/419;C07D409/12 主分类号 (IPC1-7):C07D233/64
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