发明名称 COUMPOUNDS AND METHODS FOR INHIBITING THE INTERACTION OF BCL PROTEINS WITH BINDING PARTNERS
摘要 <p>One aspect of the present invention relates to isoxazoline derivatives that bind to bcl proteins and inhibit Bcl function. Another aspect of the present invention relates to compositions comprising an isoxazoline derivative of the invention. The present invention provides methods for treating and modulating disorders associated with hyperproliferation, such as cancer.</p>
申请公布号 WO2006009869(A1) 申请公布日期 2006.01.26
申请号 WO2005US21524 申请日期 2005.06.17
申请人 INFINITY PHARMACEUTICALS, INC.;CASTRO, ALFREDO, C.;DENG, WEI;DEPEW, KRISTOPHER, M.;FOLEY, MICHAEL, A.;FRITZ, CHRISTIAN, C.;GEORGES EVANGELINOS, ASIMINA, T.;GROGAN, MICHAEL, J.;HAFEEZ, NAFEEZA;HOLSON, EDWARD, B.;HOPKINS, BRIAN, T.;KONEY, NII, O.;LIU, TAO;MANN, DAVID, A.;MARCAURELLE, LISA, A.;SNYDER, DANIEL, A.;UNDERWOOD, DENNIS, J.;WYLIE, ANDREW, A.;YU, LIN-CHEN;ZHANG, LINPING 发明人 CASTRO, ALFREDO, C.;DENG, WEI;DEPEW, KRISTOPHER, M.;FOLEY, MICHAEL, A.;FRITZ, CHRISTIAN, C.;GEORGES EVANGELINOS, ASIMINA, T.;GROGAN, MICHAEL, J.;HAFEEZ, NAFEEZA;HOLSON, EDWARD, B.;HOPKINS, BRIAN, T.;KONEY, NII, O.;LIU, TAO;MANN, DAVID, A.;MARCAURELLE, LISA, A.;SNYDER, DANIEL, A.;UNDERWOOD, DENNIS, J.;WYLIE, ANDREW, A.;YU, LIN-CHEN;ZHANG, LINPING
分类号 C07D261/02;A61K31/42;A61P35/00 主分类号 C07D261/02
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