发明名称 A PROCESS FOR THE PREPARATION OF PHENYLTETRAZOLE DERIVATIVES
摘要 <p>A process for the preparation of phenyltetrazole derivatives of formula (II) wherein R and Y are as defined in the disclosure, by direct ortho-metallation of (tetrazol-5-gammal)benzene. The compounds of formula (II) are useful intermediates for the preparation of angiotensin II antagonists.</p>
申请公布号 WO2005014560(A1) 申请公布日期 2005.02.17
申请号 WO2004EP08576 申请日期 2004.07.30
申请人 DIPHARMA S.P.A.;CASTALDI, GRAZIANO;ALLEGRINI, PIETRO;RAZZETTI, GABRIELE;BOLOGNA, ALBERTO;RASPARINI, MARCELLO;LUCCHINI, VITTORIO 发明人 CASTALDI, GRAZIANO;ALLEGRINI, PIETRO;RAZZETTI, GABRIELE;BOLOGNA, ALBERTO;RASPARINI, MARCELLO;LUCCHINI, VITTORIO
分类号 C07D257/04;C07F3/02;(IPC1-7):C07D257/04;C07F5/02 主分类号 C07D257/04
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