发明名称 |
New piperidinylamino-thieno[2,3-d] pyrimidine compounds |
摘要 |
The invention relates to 5-HT receptor antagonists. Novel piperidinylamino-thieno[2,3-d]pyrimidine compounds represented by Formula I, and synthesis and uses thereof for treating diseases mediated directly or indirectly by 5-HT receptors, are disclosed. Such conditions include central nervous system disorders such as anxiety, depression, schizophrenia, neural injury, stroke, and migraine. Methods of preparation and novel intermediates and pharmaceutical salts thereof are also included.
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申请公布号 |
US2004248904(A1) |
申请公布日期 |
2004.12.09 |
申请号 |
US20040815417 |
申请日期 |
2004.03.31 |
申请人 |
DHANOA DALE S.;BECKER OREN;NOIMAN SILVIA;REDDY SEKAR A.;CHERUKU SRINIVASA RAO;MELE'NDEZ ROSA E.;SHARADENDU ANURAG;CHEN DONGLI;MARANTZ YAEL;SHACHEM SHARON;HEIFETZ ALEXANDER;INBAL BOAZ;KESAVAN VENKITASAMY;BAR-HAIM SHAY |
发明人 |
DHANOA DALE S.;BECKER OREN;NOIMAN SILVIA;REDDY SEKAR A.;CHERUKU SRINIVASA RAO;MELE'NDEZ ROSA E.;SHARADENDU ANURAG;CHEN DONGLI;MARANTZ YAEL;SHACHEM SHARON;HEIFETZ ALEXANDER;INBAL BOAZ;KESAVAN VENKITASAMY;BAR-HAIM SHAY |
分类号 |
A61K;A61K31/519;A61P25/24;C07D;C07D495/04;C07D495/14;C07D498/02;(IPC1-7):A61K31/519 |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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