发明名称 HIGHLY PURE BASES OF 3,3-DIPHENYL PROPYLAMINE MONOESTERS
摘要 The invention relates to a compound of general formula (I) wherein A represents deuterium or hydrogen, R represents a group selected from C1-6 alkyl, C3-10 cycloalkyl or phenyl, which can be substituted by C1-3 alkoxy, fluorine, chlorine, bromine, iodine, nitro, amino, hydroxyl, oxo, mercapto o r deuterium. The C atom marked with a * (star) can be present in an (R) configuration, in an (S)-configuration or a mixture thereof. The invention i s characterised in that the above-mentioned compounds are free bases with a degree of purity of more than 97 wt %. The invention also relates to a metho d for the production of highly pure compounds of general formula (I) and to th e use thereof in the production of medicaments.
申请公布号 CA2505848(A1) 申请公布日期 2004.10.21
申请号 CA20042505848 申请日期 2004.04.03
申请人 SCHWARZ PHARMA AG 发明人 BREITENBACH, ARMIN;DREWS, ROLAND;WOLFF, HANS-MICHAEL;MEESE, CLAUS
分类号 A61K9/70;A61K31/135;A61P13/00;C07C213/10;C07C217/62;(IPC1-7):C07C217/62 主分类号 A61K9/70
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