发明名称 (CONDENSED) PYRIMIDONE AND (CONDENSED) PYRIDONE COMPOUNDS, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
摘要 Compounds of formula (I): are inhibitors of the enzyme Lp-PLA2 and are of use in therapy, in particular for treating atherosclerosis. In Formula (I) R<1>, R<2>, R<3>, R<4>, R<5>, R<6>, X and Y are as defined herein.
申请公布号 WO03087088(A3) 申请公布日期 2004.01.08
申请号 WO2003GB01550 申请日期 2003.04.10
申请人 GLAXO GROUP LIMITED;LEACH, COLIN, ANDREW;SMITH, STEPHEN, ALLAN 发明人 LEACH, COLIN, ANDREW;SMITH, STEPHEN, ALLAN
分类号 C07D215/36;A61K31/4375;A61K31/4709;A61K31/517;A61P3/10;A61P9/10;A61P19/02;A61P29/00;A61P43/00;C07D401/12;C07D403/12;C07D417/12;C07D471/04 主分类号 C07D215/36
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