发明名称 BENZYLIMIDAZOLYL SUBSTITUTED 2-QUINOLINE AND QUINAZOLINE DERIVATIVES FOR USE AS FARNESYL TRANSFERASE INHIBITORS
摘要 This invention comprises the novel compounds of formula (I) wherein r, t, Y<1>, Y<2>, R<1>, R<2>, R<3>, R<5>, R<6> and R<7> have defined meanings, having farnesyl transferase inhibiting activity; their preparation, compositions containing them and their use as a medicine to treat e.g. cancer.
申请公布号 WO03080058(A1) 申请公布日期 2003.10.02
申请号 WO2003EP02874 申请日期 2003.03.18
申请人 JANSSEN PHARMACEUTICA. N.V.;ANGIBAUD, PATRICK, RENE;VENET, MARC, GASTON;MEYER, CHRISTOPHE;BRESLIN, HENRY, JOSEPH 发明人 ANGIBAUD, PATRICK, RENE;VENET, MARC, GASTON;MEYER, CHRISTOPHE;BRESLIN, HENRY, JOSEPH
分类号 A61K31/4178;A61K31/4704;A61K31/4709;A61K31/4745;A61P1/00;A61P1/04;A61P3/04;A61P3/10;A61P5/00;A61P9/00;A61P9/10;A61P9/12;A61P11/00;A61P11/02;A61P11/06;A61P13/12;A61P15/00;A61P17/00;A61P17/04;A61P17/08;A61P17/14;A61P19/02;A61P19/06;A61P19/08;A61P25/00;A61P25/02;A61P25/28;A61P27/02;A61P29/00;A61P31/04;A61P31/12;A61P31/18;A61P33/06;A61P35/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D401/06;C07D401/14;C07D403/06;C07D471/04;C07D487/04;(IPC1-7):A61K31/470;A61K31/470;A61K31/474 主分类号 A61K31/4178
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