发明名称 METHODS FOR THE PREPARATION OF MIRTAZAPINE INTERMEDIATES
摘要 The preparation of 1-(3-carboxypyridyl-2)-4 methyl-2-phenylpiperazine dihydrate and other mirtazapine intermediates are described. These compounds are particularly useful in the preparation of mirtazapine.
申请公布号 WO02070513(A1) 申请公布日期 2002.09.12
申请号 WO2002US04340 申请日期 2002.02.14
申请人 TEVA PHARMACEUTICAL INDUSTRIES LTD.;TEVA PHARMACEUTICALS USA, INC.;METZGER, LEONID;WIZEL, SHLOMIT 发明人 METZGER, LEONID;WIZEL, SHLOMIT
分类号 A61K31/55;A61P25/24;C07D401/04;C07D471/14;C07D487/12;(IPC1-7):C07D401/04 主分类号 A61K31/55
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