发明名称 |
Phosphorous prodrugs |
摘要 |
The composition and methods of synthesis of phosphorus prodrugs are described. These methods can be used to convert negatively charged phosphorus bearing drugs into neutrally charged; lipid soluble prodrugs which are able to passively diffuse into cells and into tissues in vivo. Prodrugs for a variety of antiviral and anti-leukemic agents are described.
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申请公布号 |
US6140310(A) |
申请公布日期 |
2000.10.31 |
申请号 |
US19980073530 |
申请日期 |
1998.05.06 |
申请人 |
DRUG INNOVATION & DESIGN, INC. |
发明人 |
GLAZIER, ARNOLD |
分类号 |
C07C69/732;C07F9/24;C07F9/40;C07F9/6561;C07H19/10;C07H19/20;(IPC1-7):A61K31/70;A01N43/04;C07F9/02 |
主分类号 |
C07C69/732 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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