| 发明名称 |
METHOD FOR REDUCING IMIDATES TO PRODUCE AN 8A-AZALIDE MACROCYCLE |
| 摘要 |
A method for reducing imidate intermediates arising from Beckmann stereospecific rearrangement of a compound of general formula (II), characterized in that said intermediates are not isolated from the pyridine-based reaction medium and are directly reduced with the aid of a sufficient quantity of activated borohydride.
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| 申请公布号 |
WO0058327(A1) |
申请公布日期 |
2000.10.05 |
| 申请号 |
WO2000FR00753 |
申请日期 |
2000.03.24 |
| 申请人 |
MERIAL |
发明人 |
LEON, PATRICK;LHERMITTE, FREDERIC;LARGEAU, DENIS;GUEVEL, RONAN;PAUZE, DENIS;ODDON, GILLES |
| 分类号 |
C07H17/08;(IPC1-7):C07H17/08 |
主分类号 |
C07H17/08 |
| 代理机构 |
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