| 摘要 |
<p>PURPOSE: Provided are novel benzamidine, a production method thereof and uses thereof as competitive inhibitor of serine protease, especially, kininogenase CONSTITUTION: Provided are compounds having formula (I) wherein the radicals R, R(1),R(2), R(3), R(4), R(5) and R(6), as well as l, m, and n have the meaning indicated in the description, and the production of said compounds. The new compounds can be used to combat illness. Also described are compounds having formula (II) wherein the radicals R, R(1), R(2), R(3), R(4), R(5) and R(6), as well as l, m, and n have the meaning indicated in claim 1, and compounds having formula (III) wherein l and R have the meaning indicated in claim 1 and Y is an N protective group, or N-terminal protected or unprotected amino acid or represents H.</p> |
