发明名称 |
TRICYCLIC COMPOUNDS HAVING ACTIVITY SPECIFIC FOR INTEGRINS, PARTICULARY ALPHA-GAMA-BETA-3 INTEGRINS, METHOD FOR PREPARING SAME, INTERMEDIATES THEREFOR, USE OF SAID COMPOUNDS AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
摘要 |
Compounds of formula (I), wherein R1, R2, R3, R4, R5 and G are as defined in the description and the dotted lines indicate an optional second bond, as well as the acid, base and ester addition salts thereof, a method for preparing said compounds, intermediates therefor, the use of said compounds as drugs, and pharmaceutical compositions containing same, are disclosed. |
申请公布号 |
LT4535(B) |
申请公布日期 |
1999.08.25 |
申请号 |
LT19980000145 |
申请日期 |
1998.10.15 |
申请人 |
ROUSSEL,HOECHST MARION;GENENTECH, INC. |
发明人 |
BERNARD,SERGE;CARNIATO,DENIS;GOURVEST,JEAN-FRANCOIS;TEUTSCH,JEAN-GEORGES;KNOLLE,JOCHEN;STILZ,HANS-ULRICH;WEHNER,VOLKMAR;BODARY,SARAH C.;GADEK,THOMAS R.;MCDOWELL,ROBERT S.;PITTI,ROBERT M. |
分类号 |
B01J31/02;A61K31/00;A61K31/357;A61K31/36;A61K31/415;A61K31/4164;A61K31/4168;A61K31/505;A61P19/00;A61P19/08;A61P19/10;C07B61/00;C07C45/51;C07C45/63;C07C45/67;C07C45/71;C07C49/747;C07C49/755;C07C281/12;C07C281/18;C07C331/04;C07C331/10;C07C331/12;C07C331/14;C07C337/08;C07D233/52;C07D239/18;C07D239/42;C07D317/70 |
主分类号 |
B01J31/02 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|