发明名称 |
2-HETEROARYL-5,11-DIHYDRO-6H-DIPYRIDO[3,2-b:2',3'-e][1,4]DIA ZEPINES AND THEIR USE IN THE PREVENTION OR TREATMENT OF HIV INFECTION. |
摘要 |
Disclosed are novel 2-heteroaryl-5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]dia zepines of formula (1), wherein Z is an oxygen or sulfur atom, =NCN or a group of the formula =NOR10 wherein R10 is alkyl of 1 to 3 carbon atoms; Ar is a group of formulae (I, II, III, IV or V). These compounds are useful in the prevention or treatment of HIV infections.
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申请公布号 |
MX9603359(A) |
申请公布日期 |
1998.07.31 |
申请号 |
MX19960003359 |
申请日期 |
1996.08.13 |
申请人 |
BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. |
发明人 |
KARL D. HARGRAVE;TERENCE A. KELLY;SURESH R. KAPADIA;JOHN R. PROUDFOOT;DANIEL W. MCNEIL;USHA R. PATEL;MARIO G. CARDOZO |
分类号 |
A61K31/55;A61K31/5513;A61P31/12;A61P37/04;A61P43/00;C07D471/14;(IPC1-7):C07D471/14;C07D |
主分类号 |
A61K31/55 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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