发明名称 |
NOVEL ACYLAMINO-SUBSTITUTED ACYLANILIDE DERIVATIVES OR PHARMACEUTICAL COMPOSITION COMPRISING THE SAME |
摘要 |
Acylamino-substituted acylanilide derivatives represented by general formula (I) or salts thereof, and a pharmaceutical composition comprising the same. They have an antiandrogenic activity and are useful as a prophylactic or therapeutic agent for prostatic cancer, prostatic hypertrophy, defemination, hypertrichosis, bald head, acne, seborrhea and the like in which androgen is involved as an exacerbating factor.
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申请公布号 |
WO9822432(A1) |
申请公布日期 |
1998.05.28 |
申请号 |
WO1997JP04174 |
申请日期 |
1997.11.17 |
申请人 |
YAMANOUCHI PHARMACEUTICAL CO., LTD.;TANIGUCHI, NOBUAKI;OKADA, MINORU;KAKU, HIDETAKA;SHIMADA, ITSURO;NOZAWA, EISUKE;KOUTOKU, HIROSHI |
发明人 |
TANIGUCHI, NOBUAKI;OKADA, MINORU;KAKU, HIDETAKA;SHIMADA, ITSURO;NOZAWA, EISUKE;KOUTOKU, HIROSHI |
分类号 |
C07C255/60;C07C311/06;C07C311/13;C07C311/19;C07C311/29;C07C327/42;C07C327/48;C07D205/04;C07D207/16;C07D207/34;C07D209/08;C07D209/42;C07D211/34;C07D213/81;C07D213/82;C07D215/36;C07D215/48;C07D217/26;C07D239/28;C07D307/68;C07D309/14;C07D309/38;C07D333/34;C07D333/38;C07D333/68;C07D335/02;(IPC1-7):C07C237/22;C07C275/28;C07C335/26;C07D207/14;C07D207/48;C07D209/30;C07D209/36;C07D217/22;C07D241/12;C07D241/14;C07D307/64;C07D333/70;A61K31/165;A61K31/275;A61K31/34;A61K31/35;A61K31/38;A61K31/395;A61K31/40;A61K31/44;A61K31/47 |
主分类号 |
C07C255/60 |
代理机构 |
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代理人 |
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