发明名称 NOVEL ACYLAMINO-SUBSTITUTED ACYLANILIDE DERIVATIVES OR PHARMACEUTICAL COMPOSITION COMPRISING THE SAME
摘要 Acylamino-substituted acylanilide derivatives represented by general formula (I) or salts thereof, and a pharmaceutical composition comprising the same. They have an antiandrogenic activity and are useful as a prophylactic or therapeutic agent for prostatic cancer, prostatic hypertrophy, defemination, hypertrichosis, bald head, acne, seborrhea and the like in which androgen is involved as an exacerbating factor.
申请公布号 WO9822432(A1) 申请公布日期 1998.05.28
申请号 WO1997JP04174 申请日期 1997.11.17
申请人 YAMANOUCHI PHARMACEUTICAL CO., LTD.;TANIGUCHI, NOBUAKI;OKADA, MINORU;KAKU, HIDETAKA;SHIMADA, ITSURO;NOZAWA, EISUKE;KOUTOKU, HIROSHI 发明人 TANIGUCHI, NOBUAKI;OKADA, MINORU;KAKU, HIDETAKA;SHIMADA, ITSURO;NOZAWA, EISUKE;KOUTOKU, HIROSHI
分类号 C07C255/60;C07C311/06;C07C311/13;C07C311/19;C07C311/29;C07C327/42;C07C327/48;C07D205/04;C07D207/16;C07D207/34;C07D209/08;C07D209/42;C07D211/34;C07D213/81;C07D213/82;C07D215/36;C07D215/48;C07D217/26;C07D239/28;C07D307/68;C07D309/14;C07D309/38;C07D333/34;C07D333/38;C07D333/68;C07D335/02;(IPC1-7):C07C237/22;C07C275/28;C07C335/26;C07D207/14;C07D207/48;C07D209/30;C07D209/36;C07D217/22;C07D241/12;C07D241/14;C07D307/64;C07D333/70;A61K31/165;A61K31/275;A61K31/34;A61K31/35;A61K31/38;A61K31/395;A61K31/40;A61K31/44;A61K31/47 主分类号 C07C255/60
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