发明名称 Pharmaceutical compositions for prevention and treatment of central nervous system disorders
摘要 Patients susceptible to or suffering from central nervous system disorders (e.g., Tourette's syndrome, attention deficit disorder or schizophrenia) are treated by administering an effective amount of an aryl substituted aliphatic compound, an aryl substituted olefinic amine compound or an aryl substituted acetylenic compound. Exemplary compounds are (E)-4-(5-pyrimidinyl)-3-butene-1-amine, (E)-4-[3-(5-methoxypyridin)yl]-3-butene-1-amine, (E)-N-methyl-4-(5-pyrimidinyl)-3-butene-1-amine, (E)-N-methyl-4-[3-(5-methoxypyridin)yl]-3-butene-1-amine, (Z)-metanicotine, (E)-metanicotine, N-methyl-(3-pyridinyl)-butane-1-amine, N-methyl-4-(3-pyridinyl)-3-butyne-1-amine and (E)-N-methyl-4-[3-(6-methylpyridin)yl]-3-butene-1-amine.
申请公布号 AU4610896(A) 申请公布日期 1996.07.24
申请号 AU19960046108 申请日期 1995.12.28
申请人 R.J. REYNOLDS TOBACCO COMPANY 发明人 MEROUANE BENCHERIF;PATRICK MICHAEL LIPPIELLO;WILLIAM SCOTT CALDWELL;GARY MAURICE DULL
分类号 A61K31/44;A61K31/4406;A61K31/465;A61K31/505;A61P25/00;A61P25/16;A61P25/18;A61P25/28;C07D213/65;C07D239/26 主分类号 A61K31/44
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