发明名称 |
Balanoids |
摘要 |
A novel class of therapeutic compounds, denominated Balanoids, is disclosed. Balanoids have protein kinase C inhibitory activity and selectivity among the isoforms of protein kinase C. Balanoids are useful for treatment of diseases related to protein kinase C in animals, especially humans and is especially indicated for treatment of inflammatory diseases. |
申请公布号 |
ZA9401478(B) |
申请公布日期 |
1995.09.05 |
申请号 |
ZA19940001478 |
申请日期 |
1994.03.03 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
WILLIAM P JANZEN;CHRISTIE BOROS;ZEN-SHI LAI;YALI HALLOCK;MICHAEL PATRICK LYNCH;JULIA MARIE HEERDING;JEFFREY BAILEY NICHOLS;LAWRENCE M BALLAS;JACK B JIANG;CHRISTOPHER K BIGGERS;PHILIP F HUGHESPE;JOHN WILLIAM CROSSLEY LAMPE;STEVEN EDWARD HALL;PALANIAPPAN KULANTHAIVEL;GUNNAR ERIK JAGDMANN;HONG HU;JEAN MARIE DEFAUW;DAVID STEVEN MENALDINO;SEAN PATRICK HOLLINSHEAD |
分类号 |
C07D333/36;A61K31/165;A61K31/24;A61K31/34;A61K31/341;A61K31/38;A61K31/381;A61K31/415;A61K31/42;A61K31/425;A61K31/44;A61K31/4427;A61K31/443;A61K31/4433;A61K31/445;A61K31/4468;A61K31/495;A61K31/50;A61K31/55;A61P9/00;A61P25/00;A61P29/00;A61P31/12;A61P35/00;A61P43/00;C07C69/734;C07C233/23;C07C233/41;C07C235/48;C07C235/54;C07C235/84;C07C255/52;C07C311/09;C07C325/00;C07D207/14;C07D207/48;C07D211/56;C07D223/12;C07D257/04;C07D307/22;C07D313/04;C07D337/04;C07D401/04;C07D401/12;C07D401/14;C07D403/12;C07D403/14;C07D405/12;C07D405/14;C07D409/12;C07D413/12;C07D413/14;C07D417/12;C07D417/14;C07F9/572 |
主分类号 |
C07D333/36 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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