发明名称 RETROVIRAL PROTEASE INHIBITING COMPOUNDS, PREPARATION AND PHARMACEUTICAL
摘要 <p>A retroviral protease inhibiting compound of the formula A - X - B or a pharmaceutically acceptable salt, prodrug or ester thereof, wherein X is a linking group; A is (1) substituted amino, (2) substituted carbonyl, (3) functionalized imino, (4) functionalized alkyl, (5) functionalized acyl, (6) functionalized heterocyclic or (7) functionalized (heterocyclic)alkyl; and B is (1) substituted carbonyl independently defined as herein, (2) substituted amino independently defined as herein, (3) functionalized imino independently defined as herein, (4) functionalized alkyl independently defined as herein, (5) functionalized acyl independently defined as herein, (6) functionalized heterocyclic independently defined as herein or (7) functionalized (heterocyclic)alkyl independently defined as herein. o</p>
申请公布号 NZ233717(A) 申请公布日期 1994.02.25
申请号 NZ19900233717 申请日期 1990.05.17
申请人 ABBOTT LABORATORIES 发明人 KEMPF, DALE J;NORBECK, DANIEL W;ERICKSON, JOHN W;HING LEUNG SHAM;CODACOVI, LYNN M;PLATTNER, JACOB J
分类号 C07D295/18;A61K31/00;A61K31/10;A61K31/12;A61K31/135;A61K31/15;A61K31/165;A61K31/195;A61K31/335;A61K31/40;A61K31/415;A61K31/425;A61K31/44;A61K31/445;A61K31/47;A61K31/495;A61K31/535;A61K31/54;A61K38/00;A61P31/12;A61P37/04;C07C31/125;C07C33/18;C07C33/26;C07C33/46;C07C39/12;C07C43/164;C07C43/174;C07C43/205;C07C43/215;C07C43/23;C07C43/30;C07C43/313;C07C43/315;C07C45/00;C07C45/29;C07C45/56;C07C45/59;C07C45/62;C07C45/67;C07C45/74;C07C49/04;C07C49/12;C07C49/17;C07C49/175;C07C49/20;C07C49/215;C07C49/233;C07C49/24;C07C49/255;C07C53/134;C07C69/34;C07C69/65;C07C69/732;C07C211/27;C07C215/06;C07C215/18;C07C215/20;C07C215/28;C07C217/04;C07C225/06;C07C229/08;C07C229/26;C07C229/34;C07C233/35;C07C233/36;C07C233/40;C07C233/78;C07C235/10;C07C235/12;C07C235/34;C07C235/78;C07C237/04;C07C237/10;C07C237/20;C07C237/22;C07C239/08;C07C239/10;C07C239/18;C07C239/20;C07C247/10;C07C251/40;C07C271/20;C07C271/22;C07C271/34;C07C275/00;C07C275/16;C07C275/24;C07C311/03;C07C311/05;C07C311/06;C07C311/13;C07C311/18;C07C317/10;C07C317/28;C07C317/44;C07C323/11;C07C323/12;C07C323/25;C07C323/41;C07C323/60;C07C381/00;C07D207/06;C07D207/08;C07D207/12;C07D207/16;C07D207/24;C07D209/42;C07D211/22;C07D211/54;C07D211/62;C07D211/96;C07D213/30;C07D213/40;C07D213/42;C07D213/55;C07D213/56;C07D213/70;C07D213/81;C07D213/82;C07D215/16;C07D217/14;C07D217/16;C07D217/26;C07D231/10;C07D233/60;C07D233/61;C07D233/84;C07D239/38;C07D263/06;C07D263/32;C07D277/24;C07D277/28;C07D277/36;C07D277/42;C07D277/56;C07D279/12;C07D295/088;C07D295/14;C07D295/15;C07D295/155;C07D295/185;C07D295/20;C07D295/205;C07D295/215;C07D295/22;C07D295/26;C07D303/04;C07D303/22;C07D303/36;C07D303/48;C07D305/14;C07D307/42;C07D317/12;C07D413/12;C07D417/12;C07D487/04;C07D521/00;C07F7/02;C07F9/30;C07F9/32;C07F9/53;C07K5/02;C07K5/06;C07K5/062;C07K5/078;(IPC1-7):C07C31/125;A61K31/665;A61K31/16;A61K31/09;A61K31/085;A61K31/08;A61K31/115;A61K31/11;A61K31/045;C07F9/655;C07F9/36;C07K5/08;C07D317/02;C07D303/26;C07D303/23;C07D295/145;C07D215/18;C07D215/14;C07D211/44;C07D211/34;C07C275/18;C07C251/38;C07C247/12;C07C233/11;C07C49/11;C07C31/20;A61K37/02;A61K31/66;A61K31/505;A61K31/17;A61K31/155 主分类号 C07D295/18
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