发明名称 USE OF A NAPHTHALENMETHANAMINO DERIVATIVE AS ANTIINFLAMMATORY AGENT, WATER-SOLUBLE ACID ADDITION SALTS THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT
摘要 : USE OF A NAPHTHALENMETHANAMINO DERIVATIVE AS ANTIINFLAMMATORY AGENT, WATER-SOLUBLE ACID ADDITION SALTS THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT The compound of formula I I in free base form or in naphthalene-1,5-disulfonate acid addition salt form is known. It has now been found to possess anti-inflammatory activity. It is thus indicated for anti-inflammatory use, especially topically. Further, water-soluble acid addition salt forms have been found which are indicated for use in the preparation of e.g. pharmaceutical compositions wherein the compound is present in dissolved state in an aqueous phase.
申请公布号 CA2011247(A1) 申请公布日期 1990.09.03
申请号 CA19902011247 申请日期 1990.03.01
申请人 COOPER, PHILIP H.;MIETH, HUBERT;SCHUSTER, INGEBORG;STUETZ, ANTON;RICHTER, FRIEDRICH 发明人 COOPER, PHILIP H.;MIETH, HUBERT;SCHUSTER, INGEBORG;STUETZ, ANTON;RICHTER, FRIEDRICH
分类号 A61K31/135;A61P29/00;C07C215/54;(IPC1-7):C07C215/32 主分类号 A61K31/135
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