发明名称 PREPARATION OF AZETIDINONES
摘要 <p>Process for preparing compounds according to formula (I) <IMAGE> (I) wherein R1 and R2 represent a hydrogen atom or a protective group and R3 represents a C1-C10 alkyl or an aryl group, by oxidation of compounds according to formula (II) <IMAGE> (II) wherein R1, R2 and R3 have the above-mentioned meanings, in a two-phase system comprising: a) an organic phase including a 4-acylazetidinone compound (II) and an "onium" salt dissolved in a medium immiscible with water, b) an aqueous solution including an alkali or alkaline-earth metal salt of an organic or inorganic peracid. 4-Acyloxyazetidinones (I) are useful intermediates in the synthesis of anti-bacterial compounds.</p>
申请公布号 IL84149(D0) 申请公布日期 1988.03.31
申请号 IL19870084149 申请日期 1987.10.12
申请人 FARMITALIA CARLO ERBA S.P.A. 发明人
分类号 A61K31/397;A61P31/04;C07D205/08;(IPC1-7):C07D/ 主分类号 A61K31/397
代理机构 代理人
主权项
地址