发明名称 GUANIDINE DERIVATIVES
摘要 Compounds of formula (I): <IMAGE> (I) or a salt or acyl derivative thereof; wherein Y is either -CH=N or <IMAGE> R1 is hydroxy, halogen, (C1-4) alkyl, or (C1-4)alkoxy, R2 is a nitrogen-containing, basic substituent, R3 is hydrogen, hydroxy, halogen, (C1-4) alkyl, (C1-4) alkoxy or a nitrogen-containing, basic substituent, and R4 is hydrogen or hydroxy, are useful in treating diarrhoea and scours.
申请公布号 DE3360148(D1) 申请公布日期 1985.06.05
申请号 DE19833360148 申请日期 1983.01.25
申请人 BEECHAM GROUP PLC 发明人 NEWSOME, PETER MARTIN;BEELEY, LEE JAMES;MOSS, STEPHEN FREDERICK
分类号 A61K31/155;A61P1/12;C07C67/00;C07C201/00;C07C205/12;C07C205/26;C07C205/37;C07C205/44;C07C205/56;C07C205/58;C07C279/22;C07C281/18;(IPC1-7):C07C129/12;C07C133/12 主分类号 A61K31/155
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