发明名称 |
OLIGOPEPTIDE PRODRUGS |
摘要 |
Prodrugs are described whose structures have a oligopeptide chain which is substituted by a nucleophilic chemotherapeutic residue at the alpha -position. The products have increased cell membrane permeability and beneficial physico-chemical properties. |
申请公布号 |
ZA8302844(B) |
申请公布日期 |
1984.03.28 |
申请号 |
ZA19830002844 |
申请日期 |
1983.04.22 |
申请人 |
SMITHKLINE BECKMAN CORP |
发明人 |
GILVARG CHARLES;KINGSBURY WILLIAM DENNIS |
分类号 |
C07K1/113;A61K38/00;C07K1/20;C07K5/06;C07K5/065;C07K5/083;C07K7/06 |
主分类号 |
C07K1/113 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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