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发明名称
ANDROGEN RECEPTOR MODULATING COMPOUNDS
摘要
본 명세서에는 화학식 I의 화합물 및 약제학적으로 허용되는 이의 염 및 에스테르가 기재되어 있다. 화학식 I의 화합물은 조직-선택적 안드로겐 수용체 조절제(SARM)로서 유용성을 가지며, 전립선암 및 AR 길항작용이 요구되는 기타의 AR 의존성 상태 및 질환의 치료시에 약제로서 특히 유용하다. 화학식 I위의 화학식 I에서, R내지 R, A, B 및 E는 특허청구범위에 정의된 바와 같다.
申请公布号
KR101654529(B1)
申请公布日期
2016.09.06
申请号
KR20127013214
申请日期
2010.10.27
申请人
오리온 코포레이션
发明人
볼파르트 게르트;퇴르매캉아스 올리;살로 하리;회글룬드 이사;카르얄라이넨 아르야;크누틸라 피아;홀름 파트릭;라스쿠 시르파;베살라이넨 안니나
分类号
A61K31/4155;C07D231/14;C07D405/12
主分类号
A61K31/4155
代理机构
代理人
主权项
地址
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