发明名称 NOVEL OXAZOLIDINONE DERIVATIVE AS CETP INHIBITOR, ITS PREPARATION METHOD, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME
摘要 Disclosed are a novel oxazolidinone derivative exhibiting inhibitory activity against CETP, a preparation method thereof, and a pharmaceutical composition comprising the same. Exhibiting excellent inhibitory activity against CETP, the oxazolidinone derivative can be effectively applied to the prevention or treatment of various CETP enzyme activity- or HDL cholesterol level-related diseases such as dyslipidemia, atherosclerosis, and coronary heart disease.
申请公布号 EP2978761(A4) 申请公布日期 2016.09.07
申请号 EP20140775848 申请日期 2014.03.28
申请人 DONG-A ST CO., LTD. 发明人 PARK, JANG HYUN;SONG, SEUNG HYUN;CHUNG, HAN KOOK;KIM, HEUNG JAE;LEE, JI HYE;JANG, BYUNG JUN;KIM, EUN JUNG;JUNG, HAE HUM;RYU, CHAE LIM;HWANG, JAE-SUNG;LEE, HYUNG KI;KANG, KYUNG KOO;KIM, SOON HOE
分类号 C07D413/14;A61K31/4523;A61P3/06;A61P9/10 主分类号 C07D413/14
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