发明名称 PREPARATION OF 3,4-DIHYDRO-1,4-BENZOXAZEPIN-5(2H)-ONE DERIVATIVES BY CYCLISATION OF 2-(AM I NO ETHYLOXY) BENZOIC ACID DERIVATIVES
摘要 The present disclosure provides processes for the preparation of a compound of formula: which is a selective late sodium current inhibitor. The disclosure also provides compounds that are synthetic intermediates.
申请公布号 WO2015123519(A9) 申请公布日期 2016.11.10
申请号 WO2015US15814 申请日期 2015.02.13
申请人 GILEAD SCIENCES, INC. 发明人 CHIU, Anna;FENG, Yanshu;GAO, Hanrong;KERSCHEN, James, A.;REICHWEIN, John;SARMA, Keshab;THOMPSON, Andrew, S.;ZHAO, Xinjun
分类号 C07D267/14 主分类号 C07D267/14
代理机构 代理人
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