发明名称 ПРОИЗВОДНЫЕ АМИНОСПИРТОВ
摘要 The present invention relates to a compound formula [I]: wherein ect., X is bond, -CH2-, etc., Y is bond, -O-(CH2)n- (in which n is 1, 2, 3 or 4), etc., Z is cyano, tetrazolyl, etc., R1 is hydrogen, lower alkyl, etc., R2 is hydrogen or an amino protective group, R3 is hydrogen or lower alkyl, R4 is hydrogen or lower alkyl, R5 and R8 are each independently hydrogen, halogen, hydroxy, lower alkyl, etc., R6 is hydrogen, lower alkyl, etc., R9 is hydrogen or lower alkyl, and i is 1 or 2, or a salt thereof. The compound [I] of the present invention and pharmaceutically acceptable salts thereof are useful for the prophylactic and/or the therapeutic treatment of pollakiurea or urinary incontinence.
申请公布号 RU2005101876(A) 申请公布日期 2005.08.27
申请号 RU20050101876 申请日期 2003.06.25
申请人 ФУДЗИСАВА ФАРМАСЬЮТИКАЛ КО., ЛТД. (JP) 发明人 ХАТТОРИ Коудзи (JP);ТОМИСИТА Ясуйо (JP);ИМАНИСИ Масаси (JP)
分类号 C07D333/40;A61K31/137;A61K31/195;A61K31/235;A61K31/352;A61K31/381;A61K31/44;A61K31/4406;A61K31/455;A61K31/603;A61P13/02;A61P43/00;C07C213/00;C07C215/28;C07C215/52;C07C217/60;C07C217/92;C07C227/20;C07C229/00;C07C229/36;C07C229/38;C07C255/58;C07C269/06;C07C271/16;C07C271/22;C07C315/02;C07C317/50;C07C319/20;C07C323/32;C07C323/43;C07C323/63;C07D213/38;C07D213/40;C07D213/61;C07D213/80;C07D295/135;C07D295/155;C07D311/78 主分类号 C07D333/40
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