发明名称 HETEROCYCLIC INHIBITORS OF GLUTAMINASE
摘要 PROBLEM TO BE SOLVED: To provide methods of treating cancers, immune diseases, or neurological disorders.SOLUTION: The present invention relates to the heterocyclic compound of formula (I) further defined herein and pharmaceutical preparations thereof. The invention also relates to a method of treating cancers, immune diseases, or neurological disorders using the heterocyclic compound of the invention. The invention also relates to a pharmaceutical preparation suitable for use in a human patient, and provides a pharmaceutical preparation containing an effective amount of either of the compounds described herein (e.g. a compound of formula I, and the like), and one or more pharmaceutically acceptable excipients.SELECTED DRAWING: None
申请公布号 JP2016210810(A) 申请公布日期 2016.12.15
申请号 JP20160178240 申请日期 2016.09.13
申请人 CALITHERA BIOSCIENCES INC 发明人 JIM LI;CHEN LI-JING;BINDU GOYAL;GUY LAIDIG;TIMOTHY FRIEND STANTON;ERIC BRIAN SJOGREN
分类号 A61K31/4245;A61K31/433;A61K31/496;A61K31/501;A61K31/515;A61K31/5377;A61P25/00;A61P35/00;A61P37/00;A61P43/00;C07D271/10;C07D271/113;C07D285/12;C07D285/135;C07D417/06;C07D417/14 主分类号 A61K31/4245
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