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发明名称
AMIDATION PROCESS
摘要
This invention describes an amidation process whereby perfluorinated amino acids can be activated and treated with an amine in the presence of a coupling agent and a pyridine derivative to yield amides, without loss of optical purity.
申请公布号
EP2681188(A4)
申请公布日期
2015.04.15
申请号
EP20120777344
申请日期
2012.02.27
申请人
MERCK SHARP & DOHME CORP.
发明人
HUMPHREY, GUY
分类号
C07C231/02;C07C253/30;C07C255/46
主分类号
C07C231/02
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