发明名称 SUBSTITUTED 3-CYANOQUINOLINES AS PROTEIN TYROSINE KINASES INHIBITORS
摘要 This invention provides compounds of formula 1 wherein R 1 , G 1 , G 2 , R 4 , Z, X and n are defined herein, or a pharmaceutically acceptable salt thereof, which are useful as antineoplastic agents and in the treatment of polycystic kidney disease.
申请公布号 PT2253620(E) 申请公布日期 2014.04.15
申请号 PT20100173332T 申请日期 1999.09.22
申请人 WYETH HOLDINGS LLC 发明人 HWEI-RU TSOU;PHILIP FROST;ALLAN WISSNER;DAN MAARTEN BERGER;MIDDLETON BRAWNER FLOYD;PHILIP ROSS HAMANN;NAN ZHANG
分类号 C07D215/54;A61K31/47;A61K31/4709;A61K31/496;A61K31/5377;A61K31/541;A61K31/553;A61P13/12;A61P35/00;C07D211/00;C07D215/56;C07D317/00;C07D401/04;C07D401/12;C07D405/12;C07D409/04;C07D413/12;C07D417/12;C07D491/10;C07D491/113;C07D521/00 主分类号 C07D215/54
代理机构 代理人
主权项
地址