发明名称 |
CRYSTALLINE FORMS OF (S)-2-AMINO-3-(4-(2-AMINO-6-((R)-1-(4-CHLORO-2-(3-METHYL-1H-PYRAZOL-1-YL)PHENYL)-2,2,2-TRIFLUOROETHOXY)PYRIMIDIN-4-YL)PHENYL)PROPANOIC ACID |
摘要 |
Solid forms of (S)-2-amino-3-(4-(2-amino-6-((R)-1-(4-chloro-2-(3-methyl-1H-pyrazol-1-yl)phenyl)-2,2,2-trifluoroethoxy)pyrimidin-4-yl)phenyl)propanoic acid and salts thereof are disclosed. Pharmaceutical dosage forms and methods of their use are also disclosed. |
申请公布号 |
KR20130141572(A) |
申请公布日期 |
2013.12.26 |
申请号 |
KR20137014387 |
申请日期 |
2011.11.03 |
申请人 |
LEXICON PHARMACEUTICALS, INC. |
发明人 |
LI QUN;HU WEIFENG;YANG XIAOGEN;ZHAO JIANGQIONG;ZHAO MATTHEW MANGZHU |
分类号 |
C07D403/12;A61K31/506;A61P1/00;A61P35/00 |
主分类号 |
C07D403/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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