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发明名称
PROCESS FOR THE PREPARATION OF NEBIVOLOL
摘要
<p>The present invention relates to a novel process for the synthesis of the Nebivolol product depicted in Scheme 1, comprised of a reduced number of high-yield steps, and characterized by the enzymatic resolution of the chroman ester precursor.</p>
申请公布号
CA2818465(A1)
申请公布日期
2012.07.19
申请号
CA20112818465
申请日期
2011.11.30
申请人
MENARINI INTERNATIONAL OPERATIONS LUXEMBOURG S.A.
发明人
MAURO, SANDRO;FATTORI, DANIELA;D'ANDREA, PIERO;CIPOLLONE, AMALIA
分类号
C07D311/58
主分类号
C07D311/58
代理机构
代理人
主权项
地址
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