发明名称 |
Mutilin derivative having heterocyclic aromatic ring carboxylic acid structure in substituent at 14-position |
摘要 |
To provide a novel mutilin derivative having a substitution at the 14-position, which is a novel mutilin analogue exhibiting a potent and broad antimicrobial action against Gram-positive bacteria and Gram-negative bacteria including various drug-resistant bacteria, and which is expected to be useful as an agent for treating infectious diseases. A mutilin derivative represented by the following general formula (1): or a pharmaceutically acceptable addition salt thereof. |
申请公布号 |
US8222407(B2) |
申请公布日期 |
2012.07.17 |
申请号 |
US20080451656 |
申请日期 |
2008.05.23 |
申请人 |
FUKUDA YASUMICHI;TAKADOI MASANORI;ASAHINA YOSHIKAZU;SATO TARO;KURASAKI HARUAKI;EBISU HIROYUKI;TAKEI MASAYA;FUKUDA HIDEYUKI;KYORIN PHARMACEUTICAL CO., LTD. |
发明人 |
FUKUDA YASUMICHI;TAKADOI MASANORI;ASAHINA YOSHIKAZU;SATO TARO;KURASAKI HARUAKI;EBISU HIROYUKI;TAKEI MASAYA;FUKUDA HIDEYUKI |
分类号 |
C07D498/04;C07D401/10;C07D413/14;C07D471/04 |
主分类号 |
C07D498/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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