发明名称 Mutilin derivative having heterocyclic aromatic ring carboxylic acid structure in substituent at 14-position
摘要 To provide a novel mutilin derivative having a substitution at the 14-position, which is a novel mutilin analogue exhibiting a potent and broad antimicrobial action against Gram-positive bacteria and Gram-negative bacteria including various drug-resistant bacteria, and which is expected to be useful as an agent for treating infectious diseases. A mutilin derivative represented by the following general formula (1): or a pharmaceutically acceptable addition salt thereof.
申请公布号 US8222407(B2) 申请公布日期 2012.07.17
申请号 US20080451656 申请日期 2008.05.23
申请人 FUKUDA YASUMICHI;TAKADOI MASANORI;ASAHINA YOSHIKAZU;SATO TARO;KURASAKI HARUAKI;EBISU HIROYUKI;TAKEI MASAYA;FUKUDA HIDEYUKI;KYORIN PHARMACEUTICAL CO., LTD. 发明人 FUKUDA YASUMICHI;TAKADOI MASANORI;ASAHINA YOSHIKAZU;SATO TARO;KURASAKI HARUAKI;EBISU HIROYUKI;TAKEI MASAYA;FUKUDA HIDEYUKI
分类号 C07D498/04;C07D401/10;C07D413/14;C07D471/04 主分类号 C07D498/04
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