发明名称 |
PROCESS FOR PREPARATION OF BOSENTAN |
摘要 |
The present invention provides improved processes for preparing Bosentan. The present invention provides novel intermediates like 4,6-dihydroxy-5-(2-methoxy phenoxy)[2,2′]bipyrimidine of formula (II) and N-(6-Chloro-5-(2-ethoxyphenoxy)[2,2′-bipyrimidinyl]-4-t-butyl benzenesulfonamide cesium salt and process for preparation thereof. The invention also disclosed novel polymorphic form of the intermediates. |
申请公布号 |
EP2331513(A1) |
申请公布日期 |
2011.06.15 |
申请号 |
EP20090764309 |
申请日期 |
2009.08.07 |
申请人 |
CADILA HEALTHCARE LIMITED |
发明人 |
SATA, KAUSHILK;PANDEY, BIPIN |
分类号 |
C07D239/69;C07D239/38;C07D239/54 |
主分类号 |
C07D239/69 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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