发明名称 |
2-CYCLOAMINO-5-(PYRIDIN-4-YL)IMIDAZO[2,1-B][1,3,4]THIADIAZOLE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF |
摘要 |
The invention relates to 2-cycloamino-5-(pyridin-4-yl)imidazo[2,1-b][1,3,4]thiadiazole derivatives of the general formula (I) where: R5 is a hydrogen atom or a C1-3 alkyl, -NR7R8, or C1-3 alkyloxy group; R6 is an optionally substituted phenyl group; A is a C1-7-alklene group optionally substituted by one or two Ra groups; B is a C1-7-alkylene group optionally substituted by an Rb group; L is a nitrogen atom optionally substituted by an Rc or Rd group, or a carbon atom substituted by a Rei group and a Rd group or two Re2 groups; R7 and R8 are independently a hydrogen atom or a C1-3 alkyl group. The invention also relates to a method for preparing same and to the therapeutic use thereof. |
申请公布号 |
WO2010130934(A3) |
申请公布日期 |
2011.01.06 |
申请号 |
WO2010FR50897 |
申请日期 |
2010.05.10 |
申请人 |
SANOFI-AVENTIS;OUDOT, ROMAIN;PACAUD, CHRISTOPHE;PUECH, FREDERIC |
发明人 |
OUDOT, ROMAIN;PACAUD, CHRISTOPHE;PUECH, FREDERIC |
分类号 |
C07D513/06;A61K31/433;A61K31/4439;A61K31/496;A61P25/00;A61P29/00;A61P35/00 |
主分类号 |
C07D513/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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