发明名称 PROCESS FOR PREPARATION OF ENDOTHELIAL RECEPTOR ANTAGONIST (BOSENTAN)
摘要 <p>The present invention relates to processes for the preparation of an endothelial receptor antagonist. The present invention particularly relates to synthesis of 4-tert-butyl-N-[6-(2-hydroxyethoxy)-5-(2-methoxyphenoxy)-2-(2-pyrimidinyl)-4-pyrimidinyl] benzene sulfonamide (bosentan).</p>
申请公布号 WO2010118992(A1) 申请公布日期 2010.10.21
申请号 WO2010EP54720 申请日期 2010.04.09
申请人 SANDOZ AG;JOSHI, SHREERANG;KHAN, RASHID;BENDRE, DEVEN;SALUNKHE, DADASAHEB;GUDEKAR, SANKET 发明人 JOSHI, SHREERANG;KHAN, RASHID;BENDRE, DEVEN;SALUNKHE, DADASAHEB;GUDEKAR, SANKET
分类号 C07D403/04;A61K31/513;A61P9/12 主分类号 C07D403/04
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