发明名称 ACETYLENE DERIVATIVES HAVING HUMAN MATABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTIC ACTIVITY, PROCESS FOR PRODUCING THEM, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND USE THEREOF
摘要 The invention provides compounds of formula I wherein n, A, R, R', R'', R0, X and Y are as defined in the description, and their preparation. The compounds of formula I are useful as pharmaceuticals.
申请公布号 HU0402191(A3) 申请公布日期 2010.03.29
申请号 HU20040002191 申请日期 2002.12.03
申请人 NOVARTIS AG 发明人
分类号 C07D215/26;A61K31/32;A61K31/4035;A61K31/405;A61K31/4439;A61K31/4709;A61K31/497;A61K31/5377;A61P25/00;A61P25/04;A61P25/14;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/32;A61P25/34;A61P25/36;A61P43/00;C07C231/12;C07C233/18;C07C269/06;C07C271/16;C07D209/08;C07D209/36;C07D209/38;C07D209/44;C07D215/20;C07D401/04;C07D401/06;C07D405/04;C07D405/06;C07D405/12 主分类号 C07D215/26
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