发明名称 |
6-Substituted-2,3,4,5-Tetrahydro-1H-Benzo[d]Azepines as 5-Ht2c Receptor Agonists |
摘要 |
The present invention provides 6-substituted 2,3,4,5-tetrahydro-1H-benzo[d]azepines of Formula (I) as selective 5-HT2C receptor agonists for the treatment of 5-HT2c associated disorders including obesity, obsessive/compulsive disorder, depression, and anxiety: R6 D R?N-R''R* where R6 is -(CrC3)alkyl-S-(C0-C3)alkyl-R10, -(C1-C3)alkyl-NR11R12, -(CrC3)alkyl-O-R13. and other substituents are as defined in the specification.
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申请公布号 |
US2008255092(A1) |
申请公布日期 |
2008.10.16 |
申请号 |
US20060996457 |
申请日期 |
2006.09.01 |
申请人 |
ALLEN JOHN GORDON;BRINER KARIN;GALKA CHRISTOPHER STANLEY;HOYING RICHARD CHARLES;MARTINEZ-GRAU MARIA ANGELES;MIYASHIRO JULIE;POKROVSKAIA NATALIA;REINHARD MATTHEW ROBERT |
发明人 |
ALLEN JOHN GORDON;BRINER KARIN;GALKA CHRISTOPHER STANLEY;HOYING RICHARD CHARLES;MARTINEZ-GRAU MARIA ANGELES;MIYASHIRO JULIE;POKROVSKAIA NATALIA;REINHARD MATTHEW ROBERT |
分类号 |
A61K31/55;C07D223/16 |
主分类号 |
A61K31/55 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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