发明名称 PYRIDINE AND PYRIMIDINE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE
摘要 <p>This invention comprises the novel compounds of formula (I), wherein R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, X, Y and Z have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.</p>
申请公布号 WO2007082880(A1) 申请公布日期 2007.07.26
申请号 WO2007EP50379 申请日期 2007.01.16
申请人 JANSSEN PHARMACEUTICA N.V.;ANGIBAUD, PATRICK, RENE;VAN BRANDT, SVEN, FRANCISCUS, ANNA;MARCONNET-DECRANE, LAURENCE, FRANCOISE, BERNADETTE;ROUX, BRUNO 发明人 ANGIBAUD, PATRICK, RENE;VAN BRANDT, SVEN, FRANCISCUS, ANNA;MARCONNET-DECRANE, LAURENCE, FRANCOISE, BERNADETTE;ROUX, BRUNO
分类号 C07D239/42;A61K31/506;A61P35/00;C07D403/12;C07D405/12;C07D405/14;C07D409/12 主分类号 C07D239/42
代理机构 代理人
主权项
地址