发明名称 A PHARMACEUTICAL COMPOSITION COMPRISING AN AMIDE DERIVATIVE
摘要 <p>The present invention provides a novel modulator of the TRPV1-receptor function, comprising a compound of the formula; wherein ring A is an optionally substituted carbocycle or heterocycle, ring B is an optionally substituted benzene ring or an optionally substituted 6-membered heteroaromatic ring containing N atom, a dashed line means existence or absence of a bond, n is 1 or 2, R&lt;SUP&gt;1&lt;/SUP&gt; and R&lt;SUP&gt;2&lt;/SUP&gt; are hydrogen etc., R&lt;SUP&gt;3&lt;/SUP&gt; is lower alkyl, R&lt;SUP&gt;4&lt;/SUP&gt; is lower alkyl or aryloxy, or R&lt;SUP&gt;3&lt;/SUP&gt; and R&lt;SUP&gt;4&lt;/SUP&gt; taken together may form optionally substituted 5- or 6-membered non-aromatic heterocycle.</p>
申请公布号 WO2007069773(A1) 申请公布日期 2007.06.21
申请号 WO2006JP325313 申请日期 2006.12.13
申请人 SHIONOGI & CO., LTD.;KAI, HIROYUKI 发明人 KAI, HIROYUKI
分类号 A61K31/167;A61K31/357;A61K31/4164;A61K31/42;A61K31/421;A61K31/4245;A61K31/426;A61K31/4433;A61P25/02;A61P25/04;A61P43/00;C07C251/48;C07D233/02;C07D261/04;C07D263/06;C07D263/14;C07D271/06;C07D277/04;C07D277/10;C07D317/30;C07D319/06;C07D405/12;C07D417/04;C07D417/12 主分类号 A61K31/167
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