发明名称 Diarylsulfones as 5-HT2A antagonists
摘要 Compounds of formula I: are potent and selective antagonists of the human 5-HT<SUB>2A </SUB>receptor, and hence useful in treatment of a variety of adverse conditions of the CNS.
申请公布号 US7217740(B2) 申请公布日期 2007.05.15
申请号 US20050212789 申请日期 2005.08.26
申请人 MERCK SHARP AND DOHME 发明人 CASTRO PINEIRO JOSE LUIS;COOPER LAURA CATHERINE;GILLIGAN MYRA;HUMPHRIES ALEXANDER CHARLES;HUNT PETER ALAN;LADDUWAHETTY TAMARA;MACLEOD ANGUS MURRAY;MERCHANT KEVIN JOHN;VAN NIEL MONIQUE BODIL;WILSON KEVIN
分类号 A61K31/10;C07C317/14;C07C317/22;C07C317/24;C07C317/28;C07C317/32;C07C317/36;C07C317/42;C07C317/44;C07D205/04;C07D207/10;C07D211/38;C07D211/72;C07D213/34;C07D213/71;C07D217/24;C07D231/12;C07D233/54;C07D241/08;C07D249/08;C07D261/08;C07D271/10;C07D277/26;C07D295/096;C07D317/62;C07D319/18 主分类号 A61K31/10
代理机构 代理人
主权项
地址