发明名称 |
Diarylsulfones as 5-HT2A antagonists |
摘要 |
Compounds of formula I: are potent and selective antagonists of the human 5-HT<SUB>2A </SUB>receptor, and hence useful in treatment of a variety of adverse conditions of the CNS.
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申请公布号 |
US7217740(B2) |
申请公布日期 |
2007.05.15 |
申请号 |
US20050212789 |
申请日期 |
2005.08.26 |
申请人 |
MERCK SHARP AND DOHME |
发明人 |
CASTRO PINEIRO JOSE LUIS;COOPER LAURA CATHERINE;GILLIGAN MYRA;HUMPHRIES ALEXANDER CHARLES;HUNT PETER ALAN;LADDUWAHETTY TAMARA;MACLEOD ANGUS MURRAY;MERCHANT KEVIN JOHN;VAN NIEL MONIQUE BODIL;WILSON KEVIN |
分类号 |
A61K31/10;C07C317/14;C07C317/22;C07C317/24;C07C317/28;C07C317/32;C07C317/36;C07C317/42;C07C317/44;C07D205/04;C07D207/10;C07D211/38;C07D211/72;C07D213/34;C07D213/71;C07D217/24;C07D231/12;C07D233/54;C07D241/08;C07D249/08;C07D261/08;C07D271/10;C07D277/26;C07D295/096;C07D317/62;C07D319/18 |
主分类号 |
A61K31/10 |
代理机构 |
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